3,4-dihydropyrimidin-2(1H)-ones: Fast synthesis under microwave irradiation in solvent free conditions

被引：77

作者：

Stefani, HA ^{[1
]}

Gatti, PM ^{[1
]}

机构：

[1] Univ Sao Paulo, Fac Ciencias Farmaceut, Dept Farm, Sao Paulo, Brazil

来源：

SYNTHETIC COMMUNICATIONS | 2000年 / 30卷 / 12期

关键词：

D O I：

10.1080/00397910008087395

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Microwave irradiation has been used to accelerate the synthesis of the Biginelli compounds, in one-pot reaction between P-keto esters, aryl aldehydes, and urea. These solvent-free reactions show that it is possible to prepare these compounds in a short time reaction and with good yield and easily isolable.

引用

页码：2165 / 2173

页数：9

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