Synthesis of dihydroisoxazole nucleoside and nucleotide analogs

被引：104

作者：

Gi, HJ

Xiang, YJ

Schinazi, RF

Zhao, K

机构：

[1] NYU,DEPT CHEM,NEW YORK,NY 10003

[2] VET AFFAIRS MED CTR,GEORGIA RES CTR AIDS & HIV INFECT,DECATUR,GA 30033

[3] EMORY UNIV,SCH MED,DEPT PEDIAT,BIOCHEM PHARMACOL LAB,ATLANTA,GA 30322

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1997年 / 62卷 / 01期

关键词：

D O I：

10.1021/jo961779r

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The dihydroisoxazole nucleosides as well as their phosphonate derivatives were efiiciently prepared via 1,3-dipolar cgcloaddition reactions of nitrile oxides with corresponding vinyl nucleoside bases for antiviral studies.

引用

页码：88 / 92

页数：5

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