Mitsunobu reaction modifications allowing product isolation without chromatography: application to a small parallel library

被引：52

作者：

Pelletier, JC ^{[1
]}

Kincaid, S ^{[1
]}

机构：

[1] Wyeth Ayerst Res, Div Chem Sci, Pearl River, NY 10965 USA

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(99)02214-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Readily available reagents, triphenylphosphine resin and di-t-butylazodicarboxylate, were used in Mitsunobu reactions and the byproducts were removed without chromatography. The new modification was utilized to prepare a small, parallel, solution phase library. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：797 / 800

页数：4

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