2-azidopyrrolo[2,1-c][1,4]benzodiazepines. Synthesis of the first cyclic amidine derivatives

被引：4

作者：

Gillard, AC

Rault, S

机构：

[1] Ctr. Etud. Rech. Medicament N., U.F.R. des Sciences Pharmaceutiques, 14032 Caen, 1, rue Vaubénard

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1997年 / 34卷 / 04期

关键词：

D O I：

10.1002/jhet.5570340415

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We report the practical synthesis of the new 5-azidopyrrolo[2,1-c][1,2,4]triazolo[4,3-a][1,4]benzodiazepin-8-one and 11-alkylamino-2-azidopyrrolo[2,1-c][1,4]benzodiazepines via the corresponding hydroxy compounds.

引用

页码：1185 / 1189

页数：5

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