FTY720: a novel transplantation drug that modulates lymphocyte traffic rather than activation

被引:145
作者
Brinkmann, V
Pinschewer, D
Chiba, K
Feng, LL
机构
[1] Nova Pharma AG, Transplantat Res, CH-4002 Basel, Switzerland
[2] Univ Zurich Hosp, Inst Expt Immunol, CH-8091 Munich, Germany
[3] Yoshitorni Pharmaceut, Iruma, Saitama 358, Japan
[4] Scripps Res Inst, La Jolla, CA 92037 USA
关键词
D O I
10.1016/S0165-6147(99)01419-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:49 / 52
页数:4
相关论文
共 30 条
  • [1] DESIGN, SYNTHESIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 2-SUBSTITUTED-2-AMINO-1,3-PROPANEDIOLS - DISCOVERY OF A NOVEL IMMUNOSUPPRESSANT, FTY720
    ADACHI, K
    KOHARA, T
    NAKAO, N
    ARITA, M
    CHIBA, K
    MISHINA, T
    SASAKI, S
    FUJITA, T
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (08) : 853 - 856
  • [2] BRINKMANN V, TRANSPLANTATION, V67, pS226
  • [3] Human safety and pharmacology of FTY 720
    Brunkhorst, R
    Neumayer, HH
    Hiss, M
    Budde, K
    Lucker, P
    Mayer, T
    Brookman, L
    Schmouder, R
    [J]. TRANSPLANTATION, 1999, 67 (07) : S153 - S153
  • [4] The identification of myriocin-binding proteins
    Chen, JK
    Lane, WS
    Schreiber, SL
    [J]. CHEMISTRY & BIOLOGY, 1999, 6 (04): : 221 - 235
  • [5] Chiba K, 1996, TRANSPLANT P, V28, P1056
  • [6] Chiba K, 1998, J IMMUNOL, V160, P5037
  • [7] Induction of tolerance toward rat cardiac allografts by treatment with allochimeric class I MHC antigen and FTY720
    Chueh, SC
    Tian, L
    Wang, M
    Wang, ME
    Stepkowski, SM
    Kahan, BD
    [J]. TRANSPLANTATION, 1997, 64 (10) : 1407 - 1414
  • [8] Potent immunosuppressants, 2-alkyl-2-aminopropane-1,3-diols
    Fujita, T
    Hirose, R
    Yoneta, M
    Sasaki, S
    Inoue, K
    Kiuchi, M
    Hirase, S
    Chiba, K
    Sakamoto, H
    Arita, M
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (22) : 4451 - 4459
  • [9] SIMPLE COMPOUNDS, 2-ALKYL-2-AMINO-1,3-PROPANEDIOLS HAVE POTENT IMMUNOSUPPRESSIVE ACTIVITY
    FUJITA, T
    YONETA, M
    HIROSE, R
    SASAKI, S
    INOUE, K
    KIUCHI, M
    HIRASE, S
    ADACHI, K
    ARITA, M
    CHIBA, K
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (08) : 847 - 852
  • [10] 2-SUBSTITUTED 2-AMINOETHANOL - MINIMUM ESSENTIAL STRUCTURE FOR IMMUNOSUPPRESSIVE ACTIVITY OF ISP-I (MYRIOCIN)
    FUJITA, T
    HIROSE, R
    HAMAMICHI, N
    KITAO, Y
    SASAKI, S
    YONETA, M
    CHIBA, K
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (16) : 1857 - 1860