Iron-catalysed arylation of heteroaryl halides by Grignard reagents

被引：82

作者：

Quintin, J ^{[1
]}

Franck, X ^{[1
]}

Hocquemiller, R ^{[1
]}

Figadère, B ^{[1
]}

机构：

[1] Univ Paris Sud, CNR, BIOCIS, Lab Pharmacognosie, F-92296 Chatenay Malabry, France

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 19期

关键词：

D O I：

10.1016/S0040-4039(02)00568-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Cross-coupling reaction of phenylmagnesium bromide with heteroaryl halides, in the presence of a catalytic amount of iron salts, is reported. Yields are moderate to good, and it is worth noting that this reaction has been applied to non-activate heteroaryl halides. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：3547 / 3549

页数：3

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