Synthesis and a preliminary DNA binding study of hybrids of the carbohydrate domain of calicheamicin gamma(I)(1) and the aglycone of daunorubicin: Calichearubicins A and B

被引：31

作者：

Depew, KM

Zeman, SM

Boyer, SH

Denhart, DJ

Ikemoto, N

Danishefsky, SJ

Crothers, DM

机构：

[1] YALE UNIV,DEPT CHEM,NEW HAVEN,CT 06511

[2] COLUMBIA UNIV,DEPT CHEM,NEW YORK,NY 10027

[3] SLOAN KETTERING INST CANC RES,BIOORGAN CHEM LAB,NEW YORK,NY 10021

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1996年 / 35卷 / 23-24期

关键词：

anthracyclines; carbohydrates; DNA cleavage; drug design; total syntheses;

D O I：

10.1002/anie.199627971

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：2797 / 2801

页数：5

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