The synthesis of novel heterocyclic substituted α-amino acids;: further exploitation of α-amino acid alkynyl ketones

被引：40

作者：

Adlington, RM ^{[1
]}

Baldwin, JE ^{[1
]}

Catterick, D ^{[1
]}

Pritchard, GJ ^{[1
]}

Tang, LT ^{[1
]}

机构：

[1] Univ Oxford, Dyson Perrins Lab, Oxford OX1 3QY, England

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2000年 / 03期

关键词：

D O I：

10.1039/a909720a

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A range of novel heterocyclic substituted alpha-amino acids has been synthesised by cyclocondensations of (S)-2-tert-butoxycarbonylamino-4-oxohex-5-ynoic acid tert-butyl ester with enamines, phenylhydrazine, hydroxylamine and phenyl azide.

引用

页码：303 / 305

页数：3

共 16 条

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