Modular synthesis of isoxazolopyridones and pyrazolopyridones

被引：42

作者：

Adamo, Mauro F. A.

Duffy, Eleanor F.

Donati, Donato

Sarti-Fantoni, Piero

机构：

[1] Royal Coll Surgeons Ireland, Dept Pharmaceut & Med Chem, Ctr Synth & Chem Biol, Dublin 2, Ireland

[2] Univ Siena, Dipartimento Chim, I-53100 Siena, Italy

[3] Univ Florence, Dipartimento Chim Organ U Schiff, I-50019 Sesto Fiorentino, Italy

来源：

TETRAHEDRON | 2007年 / 63卷 / 09期

关键词：

fused isoxazoles; polyfunctional scaffold; fused pyrazoles;

D O I：

10.1016/j.tet.2006.12.044

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Herein we described the preparation of two novel heterocyclic nuclei isoxazolopyridone and pyrazolopyridone. The syntheses are modular in nature and fast to execute. The title compounds were obtained pure without intervention of chromatography. (c) 2007 Elsevier Ltd. All rights reserved.

引用

收藏

页码：2047 / 2052

页数：6

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