Parallel synthesis of benzoxazoles via microwave-assisted dielectric heating

被引：151

作者：

Pottorf, RS

Chadha, NK

Katkevics, M

Ozola, V

Suna, E

Ghane, H

Regberg, T

Player, MR

机构：

[1] Three Dimens Pharmaceut Inc, Cranbury, NJ 08512 USA

[2] Latvian Inst Organ Synth, LV-1006 Riga, Latvia

[3] Personal Chem, S-75319 Uppsala, Sweden

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 01期

关键词：

benzoxazole; microwave; parallel synthesis;

D O I：

10.1016/S0040-4039(02)02495-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A facile route to benzoxazoles has been developed using microwave-assisted dielectric heating. The ease of synthesis and workup allowed the parallel synthesis of a 48-membered library of benzoxazoles quickly and efficiently. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

收藏

页码：175 / 178

页数：4

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