Molecular pharmacology of somatostatin receptor subtypes

被引:248
作者
Patel, YC
机构
[1] MCGILL UNIV, ROYAL VICTORIA HOSP, FRASER LABS, DEPT NEUROL, MONTREAL, PQ H3A 1A1, CANADA
[2] MCGILL UNIV, ROYAL VICTORIA HOSP, FRASER LABS, DEPT NEUROSURG, MONTREAL, PQ H3A 1A1, CANADA
[3] MONTREAL NEUROL INST, MONTREAL, PQ H3A 1A1, CANADA
关键词
somatostatin; somatostatin receptor; SSTR subtypes;
D O I
10.1007/BF03350317
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:348 / 367
页数:20
相关论文
共 160 条
[51]  
HJORTH SA, 1994, J BIOL CHEM, V269, P30953
[52]   INTERNALIZATION OF THE RADIOIODINATED SOMATOSTATIN ANALOG [I-125-TYR(3)]OCTREOTIDE BY MOUSE AND HUMAN PITUITARY-TUMOR CELLS - INCREASE BY UNLABELED OCTREOTIDE [J].
HOFLAND, LJ ;
VANKOETSVELD, PM ;
WAAIJERS, M ;
ZUYDERWIJK, J ;
BREEMAN, WAP ;
LAMBERTS, SWJ .
ENDOCRINOLOGY, 1995, 136 (09) :3698-3706
[53]  
HOU CF, 1994, J BIOL CHEM, V269, P10357
[54]  
HOYER D, 1994, N-S ARCH PHARMACOL, V350, P441
[55]   Agonist-dependent regulation of cloned human somatostatin receptor types 1-5 (hSSTR1-5): Subtype selective internalization or upregulation [J].
Hukovic, N ;
Panetta, R ;
Kumar, U ;
Patel, YC .
ENDOCRINOLOGY, 1996, 137 (09) :4046-4049
[56]   SOMATOSTATIN BLOCKS A CALCIUM CURRENT IN RAT SYMPATHETIC-GANGLION NEURONS [J].
IKEDA, SR ;
SCHOFIELD, GG .
JOURNAL OF PHYSIOLOGY-LONDON, 1989, 409 :221-240
[57]   Thyroid hormone-induced expression of specific somatostatin receptor subtypes correlates with involution of the TtT-97 murine thyrotrope tumor [J].
James, RA ;
Sarapura, VD ;
Bruns, C ;
Raulf, F ;
Dowding, JM ;
Gordon, DF ;
Wood, WM ;
Ridgway, EC .
ENDOCRINOLOGY, 1997, 138 (02) :719-724
[58]   Discovery of a novel human G protein-coupled receptor gene (GPR25) located on chromosome 1 [J].
Jung, BP ;
Nguyen, T ;
Kolakowski, LF ;
Lynch, KR ;
Heng, HHQ ;
George, SR ;
ODowd, BF .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1997, 230 (01) :69-72
[59]  
KANATSUKA A, 1981, ENDOCRINOLOGY, V108, P22547
[60]   2 AMINO-ACIDS, LOCATED IN TRANSMEMBRANE DOMAIN-VI AND DOMAIN-VII, DETERMINE THE SELECTIVITY OF THE PEPTIDE AGONIST SMS-201-995 FOR THE SSTR2 SOMATOSTATIN RECEPTOR [J].
KAUPMANN, K ;
BRUNS, C ;
RAULF, F ;
WEBER, HP ;
MATTES, H ;
LUBBERT, H .
EMBO JOURNAL, 1995, 14 (04) :727-735