Molecular pharmacology of somatostatin receptor subtypes

被引:248
作者
Patel, YC
机构
[1] MCGILL UNIV, ROYAL VICTORIA HOSP, FRASER LABS, DEPT NEUROL, MONTREAL, PQ H3A 1A1, CANADA
[2] MCGILL UNIV, ROYAL VICTORIA HOSP, FRASER LABS, DEPT NEUROSURG, MONTREAL, PQ H3A 1A1, CANADA
[3] MONTREAL NEUROL INST, MONTREAL, PQ H3A 1A1, CANADA
关键词
somatostatin; somatostatin receptor; SSTR subtypes;
D O I
10.1007/BF03350317
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:348 / 367
页数:20
相关论文
共 160 条
[81]   MOLECULAR-CLONING OF A SOMATOSTATIN-28 RECEPTOR AND COMPARISON OF ITS EXPRESSION PATTERN WITH THAT OF A SOMATOSTATIN-14 RECEPTOR IN RAT-BRAIN [J].
MEYERHOF, W ;
WULFSEN, I ;
SCHONROCK, C ;
FEHR, S ;
RICHTER, D .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (21) :10267-10271
[82]   SOMATOSTATIN RECEPTOR SUBTYPE GENE-EXPRESSION IN PITUITARY-ADENOMAS [J].
MILLER, GM ;
ALEXANDER, JM ;
BIKKAL, HA ;
KATZNELSON, L ;
ZERVAS, NT ;
KLIBANSKI, A .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1995, 80 (04) :1386-1392
[83]  
MONTMINY MR, 1986, J NEUROSCI, V6, P1171
[84]   ULTRASTRUCTURAL AUTORADIOGRAPHIC LOCALIZATION OF SOMATOSTATIN-28 IN THE RAT PITUITARY-GLAND [J].
MOREL, G ;
LEROUX, P ;
PELLETIER, G .
ENDOCRINOLOGY, 1985, 116 (04) :1615-1620
[85]   ASPARTIC-ACID RESIDUE-124 IN THE THIRD TRANSMEMBRANE DOMAIN OF THE SOMATOSTATIN RECEPTOR SUBTYPE-3 IS ESSENTIAL FOR SOMATOSTATIN-14 BINDING [J].
NEHRING, RB ;
MEYERHOF, W ;
RICHTER, D .
DNA AND CELL BIOLOGY, 1995, 14 (11) :939-944
[86]  
NILSSON L, 1997, FEBS LETT, V401, P838
[87]   Differential internalization of somatostatin in COS-7 cells transfected with SST1 and SST2 receptor subtypes: A confocal microscopic study using novel fluorescent somatostatin derivatives [J].
Nouel, D ;
Gaudriault, G ;
Houle, M ;
Reisine, T ;
Vincent, JP ;
Mazella, J ;
Beaudet, A .
ENDOCRINOLOGY, 1997, 138 (01) :296-306
[88]   WIDESPREAD DISTRIBUTION OF SOMATOSTATIN RECEPTOR MESSENGER RIBONUCLEIC-ACIDS IN RAT PITUITARY [J].
OCARROLL, AM ;
KREMPELS, K .
ENDOCRINOLOGY, 1995, 136 (11) :5224-5227
[89]  
OCARROLL AM, 1992, MOL PHARMACOL, V42, P939
[90]   INHIBITION OF HUMAN BREAST-CANCER CELL (MCF-7) GROWTH-INVITRO BY THE SOMATOSTATIN ANALOG SMS 201-995 - EFFECTS ON CELL-CYCLE PARAMETERS AND APOPTOTIC CELL-DEATH [J].
PAGLIACCI, MC ;
TOGNELLINI, R ;
GRIGNANI, F ;
NICOLETTI, I .
ENDOCRINOLOGY, 1991, 129 (05) :2555-2562