Kinugasa reaction under click chemistry conditions

被引：28

作者：

Basak, A. ^{[1
]}

Chandra, K. ^{[1
]}

Pal, R. ^{[1
]}

Ghosh, S. C. ^{[1
]}

机构：

[1] Indian Inst Technol, Dept Chem, Kharagpur 721302, W Bengal, India

来源：

SYNLETT | 2007年 / 10期

关键词：

Kinugasa reaction; nitrone; beta-lactam; click chemistry;

D O I：

10.1055/s-2007-980383

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Various monocyclic beta-lactams, both cis and trans, have been successfully prepared via Kinugasa reaction mimicking the click chemistry conditions.

引用

页码：1585 / 1588

页数：4

共 37 条

[1] β-lactams as versatile synthetic intermediates for the preparation of heterocycles of biological interest [J].

Alcaide, B ;

Almendros, P .

CURRENT MEDICINAL CHEMISTRY, 2004, 11 (14) :1921-1949

[2] 4-Oxoazetidine-2-carbaldehydes as useful building blocks in stereocontrolled synthesis [J].

Alcaide, B ;

Almendros, P .

CHEMICAL SOCIETY REVIEWS, 2001, 30 (04) :226-240

[3] Synthesis of β-lactam nucleoside chimera via Kinugasa reaction and evaluation of their antibacterial activity [J].

Basak, A ;

Pal, R .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (08) :2015-2018

[4] L-proline-mediated one-pot synthesis of 3-exomethylene β-lactams via Kinugasa reaction [J].

Basak, A ;

Ghosh, SC .

SYNLETT, 2004, (09) :1637-1639

[5] An asymmetric synthesis of β-lactams:: on the use of chiral oxazolidones in the Kinugasa reaction [J].

Basak, A ;

Ghosh, SC ;

Bhowmick, T ;

Das, AK ;

Bertolasi, V .

TETRAHEDRON LETTERS, 2002, 43 (31) :5499-5501

[6]

Basak A, 2001, INDIAN J CHEM B, V40, P974

[7] An enantiospecific nitrone cycloaddition route to 3-hydroxy-2-azetidinones [J].

Basak, A ;

Bdour, HMM ;

Bhattacharya, G .

TETRAHEDRON LETTERS, 1997, 38 (14) :2535-2538

[8] PPL-catalysed hydrolysis of 3,4-disubstituted β-lactams:: Effect of chain length and stereochemistry on the enantioselectivity [J].

Basak, A ;

Bhattacharya, G ;

Bdour, HMM .

TETRAHEDRON, 1998, 54 (23) :6529-6538

[9]

BHATTHACHARYA G, 1997, THESIS INDIAN I TECH

[10] In situ click chemistry [J].

Borman, S .

CHEMICAL & ENGINEERING NEWS, 2002, 80 (06) :29-34

← 1 2 3 4 →