An efficient synthesis of tetrasubstituted cyclohexyl-1,2-diamines

被引:10
作者
Arjan, H
Boyd, E
Coumbarides, GS
Eames, J
Jones, RVH
Stenson, RA
Suggate, MJ
机构
[1] Univ London Queen Mary Coll, Dept Chem, London E1 4NS, England
[2] Syngenta, Grangemouth Mfg Ctr, Grangemouth FX3 8XG, Scotland
[3] Syngenta, Global Specialist Technol, Huddersfield HD2 1FF, W Yorkshire, England
关键词
D O I
10.1016/j.tetlet.2005.01.072
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis of symmetrically tetrasubstituted diamines derived from the (R,R)-cyclohexyl-1,2-diamine is reported. We comment on the efficiency of this sequential substitution approach as a method for the synthesis of tetrasubstituted diamines and discuss the acceptable substitution pattern for this methodology. (C) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码:1921 / 1925
页数:5
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