Stereoselective synthesis of L-733,060

被引：49

作者：

Bhaskar, G ^{[1
]}

Rao, BV ^{[1
]}

机构：

[1] Indian Inst Chem Technol, Div Organ 3, Hyderabad 500007, Andhra Pradesh, India

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 05期

关键词：

D O I：

10.1016/S0040-4039(02)02772-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Enantioselective synthesis of non-peptidic neurokinin NK1 receptor antagonist L-733,060 is described using ring-closing metathesis as a key step, starting from L-phenylglycine. (C) 2003 Elsevier Science Ltd. All rights reserved.

引用

页码：915 / 917

页数：3

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