Comprehensive survey of combinatorial library synthesis: 1999

被引:194
作者
Dolle, RE [1 ]
机构
[1] Pharmacopeia Inc, Dept Chem, Princeton, NJ 08543 USA
来源
JOURNAL OF COMBINATORIAL CHEMISTRY | 2000年 / 2卷 / 05期
关键词
D O I
10.1021/cc000055x
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:383 / 433
页数:51
相关论文
共 300 条
[71]   RXP 407, a phosphinic peptide, is a potent inhibitor of angiotensin I converting enzyme able to differentiate between its two active sites [J].
Dive, V ;
Cotton, J ;
Yiotakis, A ;
Michaud, A ;
Vassiliou, S ;
Jiracek, J ;
Vazeux, G ;
Chauvet, MT ;
Cuniasse, P ;
Corvol, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1999, 96 (08) :4330-4335
[72]   Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997 [J].
Dolle, RE .
MOLECULAR DIVERSITY, 1998, 3 (04) :199-233
[73]   Comprehensive survey of combinatorial library synthesis: 1998 [J].
Dolle, RE ;
Nelson, KH .
JOURNAL OF COMBINATORIAL CHEMISTRY, 1999, 1 (04) :235-282
[74]   Comprehensive survey of combinatorial libraries with undisclosed biological, activity: 1992-1997 [J].
Dolle, RE .
MOLECULAR DIVERSITY, 1998, 4 (04) :233-256
[75]   Parallel synthesis of prostaglandin E1 analogues [J].
Dragoli, DR ;
Thompson, LA ;
O'Brien, J ;
Ellman, JA .
JOURNAL OF COMBINATORIAL CHEMISTRY, 1999, 1 (06) :534-539
[76]   Solid-phase synthesis of irreversible human rhinovirus 3C protease inhibitors. Part 1: Optimization of tripeptides incorporating N-terminal amides [J].
Dragovich, PS ;
Zhou, R ;
Skalitzky, DJ ;
Fuhrman, SA ;
Patick, AK ;
Ford, CE ;
Meador, JW ;
Worland, ST .
BIOORGANIC & MEDICINAL CHEMISTRY, 1999, 7 (04) :589-598
[77]   Solid-phase synthesis and structural analysis of bicyclic β-turn mimetics incorporating functionality at the i to i+3 positions [J].
Eguchi, M ;
Lee, MS ;
Nakanishi, H ;
Stasiak, M ;
Lovell, S ;
Kahn, M .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1999, 121 (51) :12204-12205
[78]   Use of combinatorial and multiple parallel synthesis methodologies for the development of anti-infective natural products [J].
Fecik, RA ;
Frank, KE ;
Gentry, EJ ;
Mitscher, LA ;
Shibata, M .
PURE AND APPLIED CHEMISTRY, 1999, 71 (04) :559-564
[79]   Solid-phase SN2 macrocyclization reactions to form β-turn mimics [J].
Feng, YB ;
Pattarawarapan, M ;
Wang, ZC ;
Burgess, K .
ORGANIC LETTERS, 1999, 1 (01) :121-124
[80]   SNAr cyclizations to form cyclic peptidomimetics of β-turns [J].
Feng, YB ;
Wang, ZC ;
Jin, S ;
Burgess, K .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1998, 120 (41) :10768-10769