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Comprehensive survey of combinatorial libraries with undisclosed biological, activity: 1992-1997
被引:21
作者
:
Dolle, RE
论文数:
0
引用数:
0
h-index:
0
机构:
Pharmacopeia Inc, Dept Chem, Princeton, NJ 08345 USA
Pharmacopeia Inc, Dept Chem, Princeton, NJ 08345 USA
Dolle, RE
[
1
]
机构
:
[1]
Pharmacopeia Inc, Dept Chem, Princeton, NJ 08345 USA
来源
:
MOLECULAR DIVERSITY
|
1998年
/ 4卷
/ 04期
关键词
:
combinatorial chemistry;
heterocycle;
scaffold;
solid-phase synthesis;
solution-phase synthesis;
D O I
:
10.1023/A:1009653221320
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
[No abstract available]
引用
收藏
页码:233 / 256
页数:24
相关论文
共 252 条
[1]
A solid supported synthesis of thiol esters
[J].
Adamczyk, M
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Laboratories, Abbott Park, IL 60064, 100 Abbott Park Road
Adamczyk, M
;
Fishpaugh, JR
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Laboratories, Abbott Park, IL 60064, 100 Abbott Park Road
Fishpaugh, JR
.
TETRAHEDRON LETTERS,
1996,
37
(25)
:4305
-4308
[2]
Synthesis of 2-oxindole derivatives via the intramolecular Heck reaction on solid support
[J].
Arumugam, V
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Arumugam, V
;
Routledge, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Routledge, A
;
Abell, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Abell, C
;
论文数:
引用数:
h-index:
机构:
Balasubramanian, S
.
TETRAHEDRON LETTERS,
1997,
38
(36)
:6473
-6476
[3]
Combinatorial modification of natural products: Preparation of unencoded and encoded libraries of Rauwolfia alkaloids
[J].
Atuegbu, A
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Atuegbu, A
;
Maclean, D
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Maclean, D
;
Nguyen, C
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Nguyen, C
;
Gordon, EM
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Gordon, EM
;
Jacobs, JW
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Jacobs, JW
.
BIOORGANIC & MEDICINAL CHEMISTRY,
1996,
4
(07)
:1097
-1106
[4]
Activation method to prepare a highly reactive acylsulfonamide ''safety-catch'' linker for solid-phase synthesis
[J].
Backes, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Backes, BJ
;
Virgilio, AA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Virgilio, AA
;
Ellman, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Ellman, JA
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1996,
118
(12)
:3055
-3056
[5]
CARBON-CARBON BOND-FORMING METHODS ON SOLID SUPPORT - UTILIZATION OF KENNER SAFETY-CATCH LINKER
[J].
BACKES, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
BACKES, BJ
;
ELLMAN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
ELLMAN, JA
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1994,
116
(24)
:11171
-11172
[6]
A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries
[J].
Bailey, N
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Bailey, N
;
Dean, AW
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Dean, AW
;
Judd, DB
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Judd, DB
;
Middlemiss, D
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Middlemiss, D
;
Storer, R
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Storer, R
;
Watson, SP
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Watson, SP
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1996,
6
(12)
:1409
-1414
[7]
Baldino CM, 1997, SYNLETT, P488
[8]
Design, synthesis and use of binary encoded synthetic chemical libraries
[J].
Baldwin, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
Pharmacopeia Inc., Princeton, NJ 08540
Baldwin, JJ
.
MOLECULAR DIVERSITY,
1996,
2
(1-2)
:81
-88
[9]
SYNTHESIS OF A SMALL-MOLECULE COMBINATORIAL LIBRARY ENCODED WITH MOLECULAR TAGS
[J].
BALDWIN, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
BALDWIN, JJ
;
BURBAUM, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
BURBAUM, JJ
;
HENDERSON, I
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
HENDERSON, I
;
OHLMEYER, MHJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
OHLMEYER, MHJ
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1995,
117
(20)
:5588
-5589
[10]
A novel linkage for the solid-phase synthesis of hydroxamic acids
[J].
Bauer, U
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Bauer, U
;
Ho, WB
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Ho, WB
;
Koskinen, AMP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Koskinen, AMP
.
TETRAHEDRON LETTERS,
1997,
38
(41)
:7233
-7236
←
1
2
3
4
5
6
7
8
9
10
→
共 252 条
[1]
A solid supported synthesis of thiol esters
[J].
Adamczyk, M
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Laboratories, Abbott Park, IL 60064, 100 Abbott Park Road
Adamczyk, M
;
Fishpaugh, JR
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Laboratories, Abbott Park, IL 60064, 100 Abbott Park Road
Fishpaugh, JR
.
TETRAHEDRON LETTERS,
1996,
37
(25)
:4305
-4308
[2]
Synthesis of 2-oxindole derivatives via the intramolecular Heck reaction on solid support
[J].
Arumugam, V
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Arumugam, V
;
Routledge, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Routledge, A
;
Abell, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
UNIV CAMBRIDGE,CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND
Abell, C
;
论文数:
引用数:
h-index:
机构:
Balasubramanian, S
.
TETRAHEDRON LETTERS,
1997,
38
(36)
:6473
-6476
[3]
Combinatorial modification of natural products: Preparation of unencoded and encoded libraries of Rauwolfia alkaloids
[J].
Atuegbu, A
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Atuegbu, A
;
Maclean, D
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Maclean, D
;
Nguyen, C
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Nguyen, C
;
Gordon, EM
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Gordon, EM
;
Jacobs, JW
论文数:
0
引用数:
0
h-index:
0
机构:
AFFYMAX RES INST,SANTA CLARA,CA 95051
AFFYMAX RES INST,SANTA CLARA,CA 95051
Jacobs, JW
.
BIOORGANIC & MEDICINAL CHEMISTRY,
1996,
4
(07)
:1097
-1106
[4]
Activation method to prepare a highly reactive acylsulfonamide ''safety-catch'' linker for solid-phase synthesis
[J].
Backes, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Backes, BJ
;
Virgilio, AA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Virgilio, AA
;
Ellman, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
Ellman, JA
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1996,
118
(12)
:3055
-3056
[5]
CARBON-CARBON BOND-FORMING METHODS ON SOLID SUPPORT - UTILIZATION OF KENNER SAFETY-CATCH LINKER
[J].
BACKES, BJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
BACKES, BJ
;
ELLMAN, JA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720
ELLMAN, JA
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1994,
116
(24)
:11171
-11172
[6]
A convenient procedure for the solution phase preparation of 2-aminothiazole combinatorial libraries
[J].
Bailey, N
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Bailey, N
;
Dean, AW
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Dean, AW
;
Judd, DB
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Judd, DB
;
Middlemiss, D
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Middlemiss, D
;
Storer, R
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Storer, R
;
Watson, SP
论文数:
0
引用数:
0
h-index:
0
机构:
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
GLAXOWELLCOME MED RES CTR,STEVENAGE SG1 2NY,HERTS,ENGLAND
Watson, SP
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1996,
6
(12)
:1409
-1414
[7]
Baldino CM, 1997, SYNLETT, P488
[8]
Design, synthesis and use of binary encoded synthetic chemical libraries
[J].
Baldwin, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
Pharmacopeia Inc., Princeton, NJ 08540
Baldwin, JJ
.
MOLECULAR DIVERSITY,
1996,
2
(1-2)
:81
-88
[9]
SYNTHESIS OF A SMALL-MOLECULE COMBINATORIAL LIBRARY ENCODED WITH MOLECULAR TAGS
[J].
BALDWIN, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
BALDWIN, JJ
;
BURBAUM, JJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
BURBAUM, JJ
;
HENDERSON, I
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
HENDERSON, I
;
OHLMEYER, MHJ
论文数:
0
引用数:
0
h-index:
0
机构:
PHARMACOPEIA,PRINCETON,NJ 08540
PHARMACOPEIA,PRINCETON,NJ 08540
OHLMEYER, MHJ
.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1995,
117
(20)
:5588
-5589
[10]
A novel linkage for the solid-phase synthesis of hydroxamic acids
[J].
Bauer, U
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Bauer, U
;
Ho, WB
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Ho, WB
;
Koskinen, AMP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
UNIV OULU,DEPT CHEM,FI-90571 OULU,FINLAND
Koskinen, AMP
.
TETRAHEDRON LETTERS,
1997,
38
(41)
:7233
-7236
←
1
2
3
4
5
6
7
8
9
10
→