One-pot synthesis of polyfunctionalized cyclic urea derivatives

被引:22
作者
Fioravanti, S
Marchetti, F
Morreale, A
Pellacani, L
Tardella, PA
机构
[1] Univ Roma La Sapienza, Dipartimento Chim, I-00185 Rome, Italy
[2] Univ Pisa, Dipartimento Chim & Chim Ind, I-56124 Pisa, Italy
关键词
D O I
10.1021/ol027509e
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[GRAPHICS] Unexpectedly, imidazolidin-2-ones are easily obtained from beta-keto esters upon treatment with tert-butyl nosyloxycarbamate and calcium oxide under mild conditions. The structure of the product was established by X-ray crystallography.
引用
收藏
页码:1019 / 1021
页数:3
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