STEREOISOMERS OF APOMORPHINE DIFFER IN AFFINITY AND INTRINSIC ACTIVITY AT PRE-SYNAPTIC DOPAMINE-RECEPTORS MODULATING [H-3]DOPAMINE AND [H-3]-LABELED ACETYLCHOLINE-RELEASE IN SLICES OF CAT CAUDATE

被引:52
作者
LEHMANN, J
SMITH, RV
LANGER, SZ
机构
[1] SYNTHELABO,ETUD & RECH LABS,DEPT BIOL,58 GLACIERE,F-75621 PARIS 13,FRANCE
[2] UNIV TEXAS,COLL PHARM,INST DRUG DYNAM,AUSTIN,TX 78712
关键词
D O I
10.1016/0014-2999(83)90394-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:81 / 88
页数:8
相关论文
共 18 条
[11]  
LEHMANN J, 1982, ADV DOPAMINE RES, P25
[12]  
RIFFEE WH, 1982, ADV DOPAMINE RES
[13]   SYNTHESIS AND BIOLOGICAL-ACTIVITY OF (6AS)-10,11-DIHYDROXYAPORPHINE,OPTICAL ANTIPODE OF APOMORPHINE [J].
SAARI, WS ;
KING, SW ;
LOTTI, VJ .
JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (02) :171-172
[14]  
SEEMAN P, 1980, PHARMACOL REV, V32, P229
[15]   DOPAMINE AUTOSYNAPTIC AND POSTSYNAPTIC RECEPTORS - ELECTRO-PHYSIOLOGICAL EVIDENCE FOR DIFFERENTIAL SENSITIVITY TO DOPAMINE AGONISTS [J].
SKIRBOLL, LR ;
GRACE, AA ;
BUNNEY, BS .
SCIENCE, 1979, 206 (4414) :80-82
[16]  
SOMOGYI G, 1973, J NEUROCHEM, V19, P2667
[17]  
STARKE K, 1982, ADV PHARMACOL THER, V2, P131
[18]   SIMULTANEOUS DEMONSTRATION OF THE ACTIVATION OF PRESYNAPTIC DOPAMINE AUTORECEPTORS AND POSTSYNAPTIC DOPAMINE-RECEPTORS INVITRO BY N,N-DIPROPYL-5,6-ADTN [J].
STOOF, JC ;
HORN, AS ;
MULDER, AH .
BRAIN RESEARCH, 1980, 196 (01) :276-281