HIGH-AFFINITY BINDING-SITES FOR 1-METHYL-4-PHENYL-PYRIDINIUM ION (MPP+) ARE PRESENT IN MOUSE-BRAIN

被引:9
作者
DELZOMPO, M
BERNARDI, F
MAGGIO, R
PICCARDI, M
JOHANNESSEN, JN
CORSINI, GU
机构
[1] NINCDS,IMMUNOPHARMACOL SECT,BETHESDA,MD 20205
[2] NIMH,CLIN SCI LAB,BETHESDA,MD 20205
关键词
D O I
10.1016/0014-2999(86)90339-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:87 / 92
页数:6
相关论文
共 25 条
[1]   COMPARATIVE BEHAVIORAL, BIOCHEMICAL AND PIGMENTARY EFFECTS OF MPTP, MPP+ AND PARAQUAT IN RANA-PIPIENS [J].
BARBEAU, A ;
DALLAIRE, L ;
BUU, NT ;
POIRIER, J ;
RUCINSKA, E .
LIFE SCIENCES, 1985, 37 (16) :1529-1538
[2]   1-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE - CORRESPONDENCE OF ITS BINDING-SITES TO MONOAMINE-OXIDASE IN RAT-BRAIN, AND INHIBITION OF DOPAMINE OXIDATIVE DEAMINATION INVIVO AND INVITRO [J].
BOCCHETTA, A ;
PICCARDI, MP ;
DELZOMPO, M ;
PINTUS, S ;
CORSINI, GU .
JOURNAL OF NEUROCHEMISTRY, 1985, 45 (03) :673-676
[3]   A PRIMATE MODEL OF PARKINSONISM - SELECTIVE DESTRUCTION OF DOPAMINERGIC-NEURONS IN THE PARS COMPACTA OF THE SUBSTANTIA NIGRA BY N-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE [J].
BURNS, RS ;
CHIUEH, CC ;
MARKEY, SP ;
EBERT, MH ;
JACOBOWITZ, DM ;
KOPIN, IJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (14) :4546-4550
[4]   MECHANISM OF PARAQUAT TOXICITY IN MICE AND RATS [J].
BUS, JS ;
CAGEN, SZ ;
OLGAARD, M ;
GIBSON, JE .
TOXICOLOGY AND APPLIED PHARMACOLOGY, 1976, 35 (03) :501-513
[5]   POTENTIAL BIOACTIVATION PATHWAYS FOR THE NEUROTOXIN 1-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE (MPTP) [J].
CASTAGNOLI, N ;
CHIBA, K ;
TREVOR, AJ .
LIFE SCIENCES, 1985, 36 (03) :225-230
[6]   METABOLISM OF THE NEUROTOXIC TERTIARY AMINE, MPTP, BY BRAIN MONOAMINE-OXIDASE [J].
CHIBA, K ;
TREVOR, A ;
CASTAGNOLI, N .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 120 (02) :574-578
[7]   ACTIVE UPTAKE OF MPP+, A METABOLITE OF MPTP, BY BRAIN SYNAPTOSOMES [J].
CHIBA, K ;
TREVOR, AJ ;
CASTAGNOLI, N .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 128 (03) :1228-1232
[8]   CHRONIC PARKINSONISM SECONDARY TO INTRAVENOUS-INJECTION OF MEPERIDINE ANALOGS [J].
DAVIS, GC ;
WILLIAMS, AC ;
MARKEY, SP ;
EBERT, MH ;
CAINE, ED ;
REICHERT, CM ;
KOPIN, IJ .
PSYCHIATRY RESEARCH, 1979, 1 (03) :249-254
[9]   DEPRENYL SELECTIVELY INHIBITS [H-3] MPTP BINDING-SITES IN MONKEY BRAIN [J].
DELZOMPO, M ;
PINTUS, S ;
ZUDDAS, A ;
CORSINI, GU .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 107 (02) :285-286
[10]   INHIBITION OF [H-3] MPTP BINDING TO RAT-BRAIN BY PARGYLINE [J].
DELZOMPO, M ;
BOCCHETTA, A ;
PICCARDI, MP ;
PINTUS, S ;
CORSINI, GU .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (24) :4105-4107