EFFECT OF MEFLOQUINE ON HEPATIC DRUG-METABOLISM IN THE RAT - COMPARATIVE-STUDY WITH PRIMAQUINE

被引:22
作者
RIVIERE, JH [1 ]
BACK, DJ [1 ]
机构
[1] UNIV LIVERPOOL,DEPT PHARMACOL & THERAPEUT,POB 147,LIVERPOOL L69 3BX,ENGLAND
关键词
D O I
10.1016/0006-2952(85)90191-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:567 / 571
页数:5
相关论文
共 18 条
[1]   EFFECT OF CHLOROQUINE AND PRIMAQUINE ON ANTIPYRINE METABOLISM [J].
BACK, DJ ;
PURBA, HS ;
PARK, BK ;
WARD, SA ;
ORME, ML .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1983, 16 (05) :497-502
[2]   INHIBITION OF DRUG-METABOLISM BY THE ANTI-MALARIAL DRUGS CHLOROQUINE AND PRIMAQUINE IN THE RAT [J].
BACK, DJ ;
PURBA, HS ;
STAIGER, C ;
ORME, ML ;
BRECKENRIDGE, AM .
BIOCHEMICAL PHARMACOLOGY, 1983, 32 (02) :257-263
[3]   STUDIES ON METABOLISM OF ETHYNYLESTRADIOL IN-VITRO AND IN-VIVO - SIGNIFICANCE OF 2-HYDROXYLATION AND FORMATION OF POLAR PRODUCTS [J].
BOLT, HM ;
KAPPUS, H ;
REMMER, H .
XENOBIOTICA, 1973, 3 (12) :773-785
[4]   EFFECTS OF INSECTICIDE SYNERGISTS ON MICROSOMAL OXIDATION OF ESTRADIOL AND ETHYNYLESTRADIOL AND ON MICROSOMAL DRUG-METABOLISM [J].
BOLT, HM ;
KASSEL, H .
XENOBIOTICA, 1976, 6 (01) :33-38
[6]   MEFLOQUINE, A CLINICALLY USEFUL QUINOLINE-METHANOL ANTIMALARIAL WHICH DOES NOT SIGNIFICANTLY BIND TO DNA [J].
DAVIDSON, MW ;
GRIGGS, BG ;
BOYKIN, DW ;
WILSON, WD .
NATURE, 1975, 254 (5501) :632-634
[7]   QUANTITATIVE ASSESSMENT OF ANTI-MALARIAL ACTIVITY INVITRO BY A SEMIAUTOMATED MICRODILUTION TECHNIQUE [J].
DESJARDINS, RE ;
CANFIELD, CJ ;
HAYNES, JD ;
CHULAY, JD .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1979, 16 (06) :710-718
[8]   ADVANCES IN CHEMOTHERAPY [J].
HOWELLS, RE .
BRITISH MEDICAL BULLETIN, 1982, 38 (02) :193-199
[9]  
JENNER P, 1983, DRUG METAB DISPOS, P12
[10]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265