DOCETAXEL (TAXOTERE) DERIVATIVES - NOVEL NBCL3-BASED STEREOSELECTIVE APPROACH TO 2'-METHYLDOCETAXEL

被引：34

作者：

DENIS, JN ^{[1
]}

FKYERAT, A ^{[1
]}

GIMBERT, Y ^{[1
]}

COUTTEREZ, C ^{[1
]}

MANTELLIER, P ^{[1
]}

JOST, S ^{[1
]}

GREENE, AE ^{[1
]}

机构：

[1] UNIV GRENOBLE 1,ETUD DYNAM & STRUCT SELECT LAB,F-38041 GRENOBLE,FRANCE

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1995年 / 14期

关键词：

D O I：

10.1039/p19950001811

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The C-2 methylated 2S,3R and 2R,3S side chains of docetaxel have been enantioselectively prepared and esterified with protected 10-deacetylbaccatin III to provide novel analogues of docetaxel.

引用

页码：1811 / 1815

页数：5

共 30 条

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