BENZODIAZEPINE ANALOGS L365,260 AND L364,718 AS GASTRIN AND PANCREATIC CCK RECEPTOR ANTAGONISTS

被引：101

作者：

HUANG, SC ^{[1
]}

ZHANG, L ^{[1
]}

CHIANG, HCV ^{[1
]}

WANK, SA ^{[1
]}

MATON, PN ^{[1
]}

GARDNER, JD ^{[1
]}

JENSEN, RT ^{[1
]}

机构：

[1] NIDDKD,DIGEST DIS BRANCH,BLDG 10,ROOM 9C103,BETHESDA,MD 20892

来源：

AMERICAN JOURNAL OF PHYSIOLOGY | 1989年 / 257卷 / 01期

关键词：

D O I：

10.1152/ajpgi.1989.257.1.G169

中图分类号：

Q4 [生理学];

学科分类号：

071003 ;

摘要：

引用

页码：G169 / G174

页数：6

共 34 条

[1] RECEPTORS ON SMOOTH-MUSCLE CELLS - CHARACTERIZATION BY CONTRACTION AND SPECIFIC ANTAGONISTS [J].

BITAR, KN ;

MAKHLOUF, GM .

AMERICAN JOURNAL OF PHYSIOLOGY, 1982, 242 (04) :G400-G407

[2] BENZODIAZEPINE GASTRIN AND BRAIN CHOLECYSTOKININ RECEPTOR LIGANDS - L-365,260 [J].

BOCK, MG ;

DIPARDO, RM ;

EVANS, BE ;

RITTLE, KE ;

WHITTER, WL ;

VEBER, DF ;

ANDERSON, PS ;

FREIDINGER, RM .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (01) :13-16

[3] BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF AN EXTREMELY POTENT AND SELECTIVE NONPEPTIDE CHOLECYSTOKININ ANTAGONIST [J].

CHANG, RSL ;

LOTTI, VJ .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (13) :4923-4926

[4] A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS [J].

CHANG, RSL ;

LOTTI, VJ ;

MONAGHAN, RL ;

BIRNBAUM, J ;

STAPLEY, EO ;

GOETZ, MA ;

ALBERSSCHONBERG, G ;

PATCHETT, AA ;

LIESCH, JM ;

HENSENS, OD ;

SPRINGER, JP .

SCIENCE, 1985, 230 (4722) :177-179

[5]

CHANG RSL, 1988, NEUROL NEUROBIOL, V47, P13

[6] FUNCTIONALLY DISTINCT RECEPTORS FOR CHOLECYSTOKININ AND GASTRIN ON DISPERSED CHIEF CELLS FROM GUINEA-PIG STOMACH [J].

CHERNER, JA ;

SUTLIFF, VE ;

GRYBOWSKI, DM ;

JENSEN, RT ;

GARDNER, JD .

AMERICAN JOURNAL OF PHYSIOLOGY, 1988, 254 (02) :G151-G155

[7] CHOLECYSTOKININ-INDUCED CONTRACTION OF DISPERSED SMOOTH-MUSCLE CELLS [J].

COLLINS, SM ;

GARDNER, JD .

AMERICAN JOURNAL OF PHYSIOLOGY, 1982, 243 (06) :G497-G504

[8] RECEPTORS FOR CHOLECYSTOKININ AND GASTRIN PEPTIDES DISPLAY SPECIFIC BINDING-PROPERTIES AND ARE STRUCTURALLY DIFFERENT IN GUINEA-PIG AND DOG PANCREAS [J].

FOURMY, D ;

ZAHIDI, A ;

FABRE, R ;

GUIDET, M ;

PRADAYROL, L ;

RIBET, A .

EUROPEAN JOURNAL OF BIOCHEMISTRY, 1987, 165 (03) :683-692

[9] REGULATION OF AMYLASE RELEASE FROM DISPERSED PANCREATIC ACINAR CELLS [J].

GARDNER, JD ;

JACKSON, MJ .

JOURNAL OF PHYSIOLOGY-LONDON, 1977, 270 (02) :439-454

[10]

GARDNER JD, 1987, PHYSL GASTROINTESTIN, P1109

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