AN INTERESTING C-RING CONTRACTION IN PACLITAXEL (TAXOL(R))

被引：11

作者：

CHEN, SH

HUANG, S

ROTH, GP

机构：

[1] Bristol-Myers Squibb, Pharmaceutical Research Institute, Wallingford, CT 06492-7660

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 49期

关键词：

D O I：

10.1016/0040-4039(95)01954-G

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An interesting pinacol rearrangement involving 7-epi-6 alpha-tosylate/triflate-paclitaxel derivatives (6) and (10), with the formation of five-membered C-ring containing analogs (7) and (11), is described.

引用

页码：8933 / 8936

页数：4

共 24 条

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