A PHOTOAFFINITY INHIBITOR OF AROMATASE

被引：11

作者：

BRUEGGEMEIER, RW ^{[1
]}

SNIDER, CE ^{[1
]}

KIMBALL, JG ^{[1
]}

机构：

[1] OHIO STATE UNIV,CTR COMPREHENS CANC,COLUMBUS,OH 43210

来源：

STEROIDS | 1982年 / 40卷 / 06期

关键词：

D O I：

10.1016/0039-128X(82)90009-5

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：679 / 689

页数：11

共 22 条

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[2] INHIBITION OF PERIPHERAL AROMATIZATION BY AROMATASE INHIBITORS, 4-HYDROXY-ANDROSTENE-3,17-DIONE AND 4-ACETOXY-ANDROSTENE-3,17-DIONE [J].

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[3] AROMATASE INHIBITORS .3. STUDIES ON ANTI-FERTILITY EFFECT OF 4-ACETOXY-4-ANDROSTENE-3,17-DIONE [J].

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[5]

BRODIE AMH, 1979, J STEROID BIOCH, V10, P432

[6]

BRUEGGEMEIER RW, 1982, CANCER RES, V42, P3334

[7] SYNTHESIS AND BIOCHEMICAL EVALUATION OF INHIBITORS OF ESTROGEN BIOSYNTHESIS [J].

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FLOYD, EE ;

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JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (10) :1007-1011

[8]

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[9]

COVEY DF, 1981, J BIOL CHEM, V256, P1076

[10] ENZYME-GENERATED INTERMEDIATES DERIVED FROM 4-ANDROSTENE-3,6,17-TRIONE AND 1,4,6-ANDROSTATRIENE-3,17-DIONE CAUSE A TIME-DEPENDENT DECREASE IN HUMAN PLACENTAL AROMATASE-ACTIVITY [J].

COVEY, DF ;

HOOD, WF .

ENDOCRINOLOGY, 1981, 108 (04) :1597-1599

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