SELECTIVE REGULATION OF BETA-1-ADRENOCEPTORS AND BETA-2-ADRENOCEPTORS IN THE HUMAN-HEART BY CHRONIC BETA-ADRENOCEPTOR ANTAGONIST TREATMENT

被引:127
作者
MICHEL, MC
PINGSMANN, A
BECKERINGH, JJ
ZERKOWSKI, HR
DOETSCH, N
BRODDE, OE
机构
[1] UNIV ESSEN GESAMTHSCH,DIV RENAL & HYPERTENS DIS,MED KLIN & POLIKLIN,BIOCHEM RES LAB,D-4300 ESSEN 1,FED REP GER
[2] UNIV ESSEN GESAMTHSCH,DIV THORAC & CARDIOVASC SURG,D-4300 ESSEN 1,FED REP GER
关键词
D O I
10.1111/j.1476-5381.1988.tb11576.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:685 / 692
页数:8
相关论文
共 37 条
[1]   ELEVATION OF BETA-ADRENERGIC-RECEPTOR DENSITY IN HUMAN-LYMPHOCYTES AFTER PROPRANOLOL ADMINISTRATION [J].
AARONS, RD ;
NIES, AS ;
GAL, J ;
HEGSTRAND, LR ;
MOLINOFF, PB .
JOURNAL OF CLINICAL INVESTIGATION, 1980, 65 (05) :949-957
[2]  
AARONS RD, 1982, J PHARMACOL EXP THER, V221, P439
[3]   THE PHARMACOLOGY OF A BETA-2-SELECTIVE ADRENOCEPTOR ANTAGONIST (ICI-118,551) [J].
BILSKI, AJ ;
HALLIDAY, SE ;
FITZ GERALD, JD ;
WALE, JL .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1983, 5 (03) :430-437
[4]  
BOYUM A, 1968, SCAND J CLIN LAB INV, VS 21, P77
[5]   BETA-ADRENERGIC FUNCTION IN HEART-MUSCLE DISEASE AND HEART-FAILURE [J].
BRISTOW, MR ;
KANTROWITZ, NE ;
GINSBURG, R ;
FOWLER, MB .
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 1985, 17 :41-52
[6]   BETA-1-ADRENERGIC-RECEPTOR AND BETA-2-ADRENERGIC-RECEPTOR SUBPOPULATIONS IN NONFAILING AND FAILING HUMAN VENTRICULAR MYOCARDIUM - COUPLING OF BOTH RECEPTOR SUBTYPES TO MUSCLE-CONTRACTION AND SELECTIVE BETA-1-RECEPTOR DOWN-REGULATION IN HEART-FAILURE- [J].
BRISTOW, MR ;
GINSBURG, R ;
UMANS, V ;
FOWLER, M ;
MINOBE, W ;
RASMUSSEN, R ;
ZERA, P ;
MENLOVE, R ;
SHAH, P ;
JAMIESON, S ;
STINSON, EB .
CIRCULATION RESEARCH, 1986, 59 (03) :297-309
[7]   DECREASED CATECHOLAMINE SENSITIVITY AND BETA-ADRENERGIC-RECEPTOR DENSITY IN FAILING HUMAN HEARTS [J].
BRISTOW, MR ;
GINSBURG, R ;
MINOBE, W ;
CUBICCIOTTI, RS ;
SAGEMAN, WS ;
LURIE, K ;
BILLINGHAM, ME ;
HARRISON, DC ;
STINSON, EB .
NEW ENGLAND JOURNAL OF MEDICINE, 1982, 307 (04) :205-211
[8]  
BRODDE OE, 1984, J CARDIOVASC PHARM, V6, P1184
[9]   EFFECTS OF BETA-ADRENOCEPTOR ANTAGONIST ADMINISTRATION ON BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - THE ROLE OF THE INTRINSIC SYMPATHOMIMETIC ACTIVITY [J].
BRODDE, OE ;
DAUL, A ;
STUKA, N ;
OHARA, N ;
BORCHARD, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 328 (04) :417-422
[10]  
BRODDE OE, 1987, ISI ATLAS-PHARMACOL, V1, P107