SELECTIVE REGULATION OF BETA-1-ADRENOCEPTORS AND BETA-2-ADRENOCEPTORS IN THE HUMAN-HEART BY CHRONIC BETA-ADRENOCEPTOR ANTAGONIST TREATMENT

被引:127
作者
MICHEL, MC
PINGSMANN, A
BECKERINGH, JJ
ZERKOWSKI, HR
DOETSCH, N
BRODDE, OE
机构
[1] UNIV ESSEN GESAMTHSCH,DIV RENAL & HYPERTENS DIS,MED KLIN & POLIKLIN,BIOCHEM RES LAB,D-4300 ESSEN 1,FED REP GER
[2] UNIV ESSEN GESAMTHSCH,DIV THORAC & CARDIOVASC SURG,D-4300 ESSEN 1,FED REP GER
关键词
D O I
10.1111/j.1476-5381.1988.tb11576.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:685 / 692
页数:8
相关论文
共 37 条
[11]   REGIONAL DISTRIBUTION OF BETA-ADRENOCEPTORS IN THE HUMAN-HEART - COEXISTENCE OF FUNCTIONAL BETA-1-ADRENOCEPTOR AND BETA-2-ADRENOCEPTOR IN BOTH ATRIA AND VENTRICLES IN SEVERE CONGESTIVE CARDIOMYOPATHY [J].
BRODDE, OE ;
SCHULER, S ;
KRETSCH, R ;
BRINKMANN, M ;
BORST, HG ;
HETZER, R ;
REIDEMEISTER, JC ;
WARNECKE, H ;
ZERKOWSKI, HR .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1986, 8 (06) :1235-1242
[12]   HUMAN-HEART BETA-ADRENOCEPTORS - A FAIR COMPARISON WITH LYMPHOCYTE BETA-ADRENOCEPTORS [J].
BRODDE, OE ;
BECKERINGH, JJ ;
MICHEL, MC .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1987, 8 (10) :403-407
[13]   BETA-ADRENOCEPTOR ANTAGONISTS (NONSELECTIVE AS WELL AS BETA-1-SELECTIVE) WITH PARTIAL AGONISTIC ACTIVITY DECREASE BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - EVIDENCE FOR A BETA-2-AGONISTIC COMPONENT OF THE PARTIAL AGONISTIC ACTIVIT [J].
BRODDE, OE ;
SCHEMUTH, R ;
BRINKMANN, M ;
WANG, XL ;
DAUL, A ;
BORCHARD, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 333 (02) :130-138
[14]  
BRODDE OE, 1986, J CARDIOVASC PHARM, V8, pS29
[15]   DIFFERENTIATION OF BETA-1-ADRENOCEPTOR AND BETA-2-ADRENOCEPTOR-MEDIATED EFFECTS IN HUMANS [J].
BRODDE, OE ;
DAUL, A ;
WELLSTEIN, A ;
PALM, D ;
MICHEL, MC ;
BECKERINGH, JJ .
AMERICAN JOURNAL OF PHYSIOLOGY, 1988, 254 (02) :H199-H206
[16]   TERBUTALINE-INDUCED DESENSITIZATION OF HUMAN-LYMPHOCYTE BETA-2-ADRENOCEPTORS - ACCELERATED RESTORATION OF BETA-ADRENOCEPTOR RESPONSIVENESS BY PREDNISONE AND KETOTIFEN [J].
BRODDE, OE ;
BRINKMANN, M ;
SCHEMUTH, R ;
OHARA, N ;
DAUL, A .
JOURNAL OF CLINICAL INVESTIGATION, 1985, 76 (03) :1096-1101
[17]   AUGMENTATION OF PLASMA NOR-EPINEPHRINE RESPONSE TO EXERCISE IN PATIENTS WITH CONGESTIVE HEART FAILURE [J].
CHIDSEY, CA ;
BRAUNWALD, E ;
HARRISON, DC .
NEW ENGLAND JOURNAL OF MEDICINE, 1962, 267 (13) :650-&
[18]   PLASMA NOREPINEPHRINE AS A GUIDE TO PROGNOSIS IN PATIENTS WITH CHRONIC CONGESTIVE HEART-FAILURE [J].
COHN, JN ;
LEVINE, TB ;
OLIVARI, MT ;
GARBERG, V ;
LURA, D ;
FRANCIS, GS ;
SIMON, AB ;
RECTOR, T .
NEW ENGLAND JOURNAL OF MEDICINE, 1984, 311 (13) :819-823
[19]   RATIONALE FOR BETA-ADRENERGIC BLOCKING-DRUGS IN CARDIOMYOPATHY [J].
FOWLER, MB ;
BRISTOW, MR .
AMERICAN JOURNAL OF CARDIOLOGY, 1985, 55 (10) :D120-D124
[20]   RESPONSE OF PLASMA NOREPINEPHRINE AND EPINEPHRINE TO DYNAMIC EXERCISE IN PATIENTS WITH CONGESTIVE HEART-FAILURE [J].
FRANCIS, GS ;
GOLDSMITH, SR ;
ZIESCHE, SM ;
COHN, JN .
AMERICAN JOURNAL OF CARDIOLOGY, 1982, 49 (05) :1152-1156