EFFECTS INVITRO OF MEDROXYPROGESTERONE ACETATE ON STEROID METABOLIZING ENZYMES IN THE RAT - SELECTIVE-INHIBITION OF 3-ALPHA-HYDROXYSTEROID OXIDOREDUCTASE ACTIVITY

被引:13
作者
SUNDE, A [1 ]
ROSNESS, PA [1 ]
EIKNES, KB [1 ]
机构
[1] UNIV TRONDHEIM,INST BIOPHYS,N-7034 TRONDHEIM,NORWAY
关键词
D O I
10.1016/0022-4731(82)90122-4
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:197 / 203
页数:7
相关论文
共 31 条
[21]   INVITRO [7-H-3]-TESTOSTERONE METABOLISM BY RAT VENTRAL PROSTATE - EFFECT OF SOME EXOGENOUS COMPOUNDS [J].
PATWARDHAN, VV ;
LANTHIER, A .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1975, 6 (02) :137-141
[22]   PRODUCTION AND EFFECTS OF 7ALPHA-HYDROXYTESTOSTERONE ON TESTOSTERONE AND DIHYDROTESTOSTERONE METABOLISM IN RAT TESTIS [J].
ROSNESS, PA ;
SUNDE, A ;
EIKNES, KB .
BIOCHIMICA ET BIOPHYSICA ACTA, 1977, 488 (01) :55-68
[23]   INFLUENCE OF MEDROXYPROGESTERONEACETATE ON TESTOSTERONE METABOLISM BY CULTURED HUMAN FIBROBLASTS - MODEL FOR DRUG-STEROID INTERACTION [J].
SAENGER, P ;
SHANIES, DD ;
NEW, MI .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1973, 37 (05) :760-764
[24]  
SANCHEZ FA, 1979, INT J ANDROL, V2, P136
[25]   METABOLISM OF 5-ALPHA-ANDROSTANE-3-BETA,17-BETA-DIOL TO 17-BETA-HYDROXY-5-ALPHA-ANDROSTAN-3-ONE AND 5-ALPHA-ANDROSTAN-3-ALPHA,17-BETA-DIOL IN THE RAT [J].
SUNDE, A ;
ROSNESS, PA ;
EIKNES, KB .
BIOCHIMICA ET BIOPHYSICA ACTA, 1979, 574 (02) :240-247
[26]   SEPARATION OF EPIMERIC 3-HYDROXYANDROSTANES AND 3-HYDROXYANDROSTENES BY THIN-LAYER CHROMATOGRAPHY ON SILICA-GEL [J].
SUNDE, A ;
STENSTAD, P ;
EIKNES, KB .
JOURNAL OF CHROMATOGRAPHY, 1979, 175 (01) :219-221
[27]   ANDROGENIC CONTROL OF MICROSOMAL 3-ALPHA-HYDROXYSTEROID OXIDOREDUCTASES IN RAT-KIDNEY [J].
VERHOEVEN, G ;
DEMOOR, P .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1977, 8 (02) :113-119
[28]   EFFECTS OF ANDROSTANES, 5-ALPHA-ANDROSTANES, 5-BETA-ANDROSTANES, ESTRENES AND ESTRATRIENES ON SERUM GONADOTROPIN LEVELS AND VENTRAL PROSTATE WEIGHTS IN GONADECTOMIZED, ADULT MALE RATS [J].
VERJANS, HL ;
EIKNES, KB .
ACTA ENDOCRINOLOGICA, 1976, 83 (01) :201-210
[29]   CELLULAR REGULATION OF METABOLISM OF ANDROGENS IN RAT ORAL-MUCOSA .1. EFFECT OF MEDROXYPROGESTERONE ACETATE (MPA) ON SOLUBLE SUPERNATANT (CYTOSOL) ACTIVATING MICROSOMAL DELTA-4-3-KETOSTEROID-5 ALPHA-REDUCTASE AND 17BETA-HYDROXYSTEROID OXIDOREDUCTASE ENZYME-SYSTEMS [J].
VITTEK, J ;
RAPPAPORT, SC ;
SOUTHREN, AL ;
GORDON, GG .
JOURNAL OF DENTAL RESEARCH, 1978, 57 (11-1) :1016-1018
[30]   EFFECT OF PROGESTINS ON ANDROGEN DELTA-4-3-KETOSTEROID-5 ALPHA-A-RING REDUCTASE SYSTEM IN RAT ORAL-MUCOSA [J].
VITTEK, J ;
ALTMAN, K ;
RAPPAPORT, SC ;
GORDON, GG ;
HAGEDORN, J ;
SOUTHREN, AL .
JOURNAL OF DENTAL RESEARCH, 1978, 57 (03) :511-519