SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF A SERIES OF AMINOPYRIDAZINE DERIVATIVES OF GAMMA-AMINOBUTYRIC-ACID ACTING AS SELECTIVE GABA-A ANTAGONISTS

被引：97

作者：

WERMUTH, CG ^{[1
]}

BOURGUIGNON, JJ ^{[1
]}

SCHLEWER, G ^{[1
]}

GIES, JP ^{[1
]}

SCHOENFELDER, A ^{[1
]}

MELIKIAN, A ^{[1
]}

BOUCHET, MJ ^{[1
]}

CHANTREUX, D ^{[1
]}

MOLIMARD, JC ^{[1
]}

HEAULME, M ^{[1
]}

CHAMBON, JP ^{[1
]}

BIZIERE, K ^{[1
]}

机构：

[1] GRP SANOFI,CTR RECH CLIN MIDY,F-34082 MONTPELLIER,FRANCE

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 02期

关键词：

D O I：

10.1021/jm00385a003

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：239 / 249

页数：11

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