CRYSTAL-STRUCTURES OF ALPHA-FUNALTREXAMINE AND BETA-FUNALTREXAMINE - CONFORMATIONAL REQUIREMENT OF THE FUMARAMATE MOIETY IN THE IRREVERSIBLE BLOCKAGE OF MU-OPIOID RECEPTORS

被引：28

作者：

GRIFFIN, JF ^{[1
]}

LARSON, DL ^{[1
]}

PORTOGHESE, PS ^{[1
]}

机构：

[1] UNIV MINNESOTA,COLL PHARM,DEPT MED CHEM,MINNEAPOLIS,MN 55455

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 05期

关键词：

D O I：

10.1021/jm00155a031

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：778 / 783

页数：6

共 23 条

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[17] CRYSTAL-STRUCTURE OF A NARCOTIC ANALGESIC - OXYMORPHONE HYDRATE
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[18] TAKEMORI AE, 1985, ANNU REV PHARMACOL, V25, P193
[19] TAKEMORI AE, 1981, EUR J PHARMACOL, V70, P445, DOI 10.1016/0014-2999(81)90355-1
[20] IMPROVED ASSAYS FOR THE ASSESSMENT OF KAPPA-PROPERTIES AND DELTA-PROPERTIES OF OPIOID LIGANDS
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[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 85 (02) : 163 - 170

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