STEREOSELECTIVE SYNTHESES OF THE 14-HYDROXY EPIMERS OF AMPHOTERICIN-B METHYL-ESTER

被引：8

作者：

COSTELLO, BJ ^{[1
]}

DRIVER, MJ ^{[1
]}

MACLACHLAN, WS ^{[1
]}

TAYLOR, AW ^{[1
]}

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT,YEW TREE BOTTOM RD,EPSOM KT18 5XQ,SURREY,ENGLAND

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1993年 / 16期

关键词：

D O I：

10.1039/p19930001829

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

(14R)-Hydroxyamphotericin B methyl ester 8 and its (14S)-epimer 12 have been obtained by way of m-CPBA oxidation of the enol ethers 5 and 6 respectively.

引用

页码：1829 / 1830

页数：2

共 21 条

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