A NEW FACILE SYNTHESIS OF A THROMBOXANE B-2 PRECURSOR

被引：5

作者：

BOOYSEN, JF ^{[1
]}

HOLZAPFEL, CW ^{[1
]}

机构：

[1] RAND AFRIKAANS UNIV,DEPT CHEM & BIOCHEM,JOHANNESBURG 2000,SOUTH AFRICA

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 10期

关键词：

D O I：

10.1080/00397919508011758

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A short, stereocontrolled synthesis of a key intermediate in the synthesis of thromboxane B-2 is described. The approach is based on the use of N,N-diethyl(phenylsulfonyl)acetamide as nucleophile in a palladium-catalysed nucleophilic substitution reaction.

引用

页码：1461 / 1472

页数：12

共 11 条

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