MECHANISMS OF GROWTH-INHIBITION BY NONSTEROIDAL ANTIESTROGENS IN HUMAN-BREAST CANCER-CELLS

被引:72
作者
SUTHERLAND, RL [1 ]
WATTS, CKW [1 ]
HALL, RE [1 ]
RUENITZ, PC [1 ]
机构
[1] UNIV GEORGIA, COLL PHARM, ATHENS, GA 30602 USA
关键词
D O I
10.1016/0022-4731(87)90165-8
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:891 / 897
页数:7
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共 32 条
[21]  
RUENITZ PC, 1984, DRUG METAB DISPOS, V12, P478
[22]   SUBSTITUTED-VINYL HYDROXYTRIARYLETHYLENES, 1-[4-[2-(DIETHYLAMINO)ETHOXY]PHENYL]-1-(4-HYDROXYPHENYL)-2-PHENYLETHYLENES - SYNTHESIS AND EFFECTS ON MCF-7 BREAST-CANCER CELL-PROLIFERATION [J].
RUENITZ, PC ;
BAGLEY, JR ;
WATTS, CKW ;
HALL, RE ;
SUTHERLAND, RL .
JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (12) :2511-2519
[23]   METABOLISM OF CLOMIPHENE IN THE RAT - ESTROGEN-RECEPTOR AFFINITY AND ANTIESTROGENIC ACTIVITY OF CLOMIPHENE METABOLITES [J].
RUENITZ, PC ;
BAGLEY, JR ;
MOKLER, CM .
BIOCHEMICAL PHARMACOLOGY, 1983, 32 (19) :2941-2947
[24]   TAMOXIFEN INDUCES ACCUMULATION OF MCF-7 HUMAN MAMMARY-CARCINOMA CELLS IN THE G0-G1 PHASE OF THE CELL-CYCLE [J].
SUTHERLAND, RL ;
GREEN, MD ;
HALL, RE ;
REDDEL, RR ;
TAYLOR, IW .
EUROPEAN JOURNAL OF CANCER & CLINICAL ONCOLOGY, 1983, 19 (05) :615-621
[25]   HIGH-AFFINITY ANTI-ESTROGEN BINDING-SITE DISTINCT FROM THE ESTROGEN-RECEPTOR [J].
SUTHERLAND, RL ;
MURPHY, LC ;
FOO, MS ;
GREEN, MD ;
WHYBOURNE, AM .
NATURE, 1980, 288 (5788) :273-275
[26]   DEFINITION OF 2 DISTINCT MECHANISMS OF ACTION OF ANTIESTROGENS ON HUMAN-BREAST CANCER CELL-PROLIFERATION USING HYDROXYTRIPHENYLETHYLENES WITH HIGH-AFFINITY FOR THE ESTROGEN-RECEPTOR [J].
SUTHERLAND, RL ;
WATTS, CKW ;
RUENITZ, PC .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1986, 140 (02) :523-529
[27]  
SUTHERLAND RL, 1983, CANCER RES, V43, P3998
[28]  
SUTHERLAND RL, 1984, PROGR CANCER RES THE, V31, P193
[29]  
TAYLOR IW, 1983, CANCER RES, V43, P4007
[30]   MICROSOMAL BINDING-SITES FOR ANTIESTROGENS IN RAT-LIVER - PROPERTIES AND DETERGENT SOLUBILIZATION [J].
WATTS, CKW ;
SUTHERLAND, RL .
BIOCHEMICAL JOURNAL, 1986, 236 (03) :903-911