EFFECTIVE BLOCKING OF HIV-1 PROTEINASE ACTIVITY BY CHARACTERISTIC INHIBITORS OF ASPARTIC PROTEINASES

被引:167
作者
RICHARDS, AD
ROBERTS, R
DUNN, BM
GRAVES, MC
KAY, J
机构
[1] UNIV WALES COLL CARDIFF,DEPT BIOCHEM,POB 903,CARDIFF CF1 1ST,WALES
[2] UNIV FLORIDA,J HILLIS MILLER HLTH CTR,DEPT BIOCHEM & MOLEC BIOL,GAINESVILLE,FL 32610
[3] HOFFMANN LA ROCHE INC,ROCHE RES CTR,DEPT MOLEC GENET,NUTLEY,NJ 07110
关键词
D O I
10.1016/0014-5793(89)81251-7
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:113 / 117
页数:5
相关论文
共 22 条
  • [1] 2-STEP AFFINITY-CHROMATOGRAPHIC PURIFICATION OF CATHEPSIN-D FROM PIG MYOMETRIUM WITH HIGH-YIELD
    AFTING, EG
    BECKER, ML
    [J]. BIOCHEMICAL JOURNAL, 1981, 197 (02) : 519 - 522
  • [2] BILLICH S, 1988, J BIOL CHEM, V263, P17905
  • [3] ON THE RATIONAL DESIGN OF RENIN INHIBITORS - X-RAY STUDIES OF ASPARTIC PROTEINASES COMPLEXED WITH TRANSITION-STATE ANALOGS
    BLUNDELL, TL
    COOPER, J
    FOUNDLING, SI
    JONES, DM
    ATRASH, B
    SZELKE, M
    [J]. BIOCHEMISTRY, 1987, 26 (18) : 5585 - 5590
  • [4] THE PH-DEPENDENCE OF THE HYDROLYSIS OF CHROMOGENIC SUBSTRATES OF THE TYPE, LYS-PRO-XAA-YAA-PHE-(NO2)PHE-ARG-LEU, BY SELECTED ASPARTIC PROTEINASES - EVIDENCE FOR SPECIFIC INTERACTIONS IN SUBSITES S3 AND S2
    DUNN, BM
    VALLER, MJ
    ROLPH, CE
    FOUNDLING, SI
    JIMENEZ, M
    KAY, J
    [J]. BIOCHIMICA ET BIOPHYSICA ACTA, 1987, 913 (02) : 122 - 130
  • [5] ELLIS KJ, 1982, METHOD ENZYMOL, V87, P405
  • [6] GIAM CZ, 1988, J BIOL CHEM, V263, P14617
  • [7] AN 11-KDA FORM OF HUMAN IMMUNODEFICIENCY VIRUS PROTEASE EXPRESSED IN ESCHERICHIA-COLI IS SUFFICIENT FOR ENZYMATIC-ACTIVITY
    GRAVES, MC
    LIM, JJ
    HEIMER, EP
    KRAMER, RA
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1988, 85 (08) : 2449 - 2453
  • [8] PARTIAL-PURIFICATION AND SUBSTRATE ANALYSIS OF BACTERIALLY EXPRESSED HIV PROTEASE BY MEANS OF MONOCLONAL-ANTIBODY
    HANSEN, J
    BILLICH, S
    SCHULZE, T
    SUKROW, S
    MOELLING, K
    [J]. EMBO JOURNAL, 1988, 7 (06) : 1785 - 1791
  • [9] THE EFFECTS OF LACTOYL-PEPSTATIN AND THE PEPSIN INHIBITOR PEPTIDE ON PIG CATHEPSIN-D
    KAY, J
    AFTING, EG
    AOYAGI, T
    DUNN, BM
    [J]. BIOCHEMICAL JOURNAL, 1982, 203 (03) : 795 - 797
  • [10] INTERACTION OF HUMAN CATHEPSIN-D WITH INHIBITOR PEPSTATIN
    KNIGHT, CG
    BARRETT, AJ
    [J]. BIOCHEMICAL JOURNAL, 1976, 155 (01) : 117 - 125