BIPHASIC COMPETITION BETWEEN OPIATES AND ENKEPHALINS - DOES IT INDICATE THE EXISTENCE OF A COMMON HIGH-AFFINITY (MU-1) BINDING-SITE

被引:8
作者
SARNE, Y
KENNER, A
机构
关键词
D O I
10.1016/0024-3205(87)90407-3
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:555 / 562
页数:8
相关论文
共 17 条
[1]   EVALUATION OF THE INTERACTIONS OF MU AND DELTA SELECTIVE LIGANDS WITH [H-3]D-ALA2-D-LEU5-ENKEPHALIN BINDING TO MOUSE-BRAIN MEMBRANES [J].
BARRETT, RW ;
VAUGHT, JL .
LIFE SCIENCES, 1983, 33 (24) :2439-2448
[2]   INTERCONVERTING MU-FORMS AND DELTA-FORMS OF THE OPIATE RECEPTOR IN RAT STRIATAL PATCHES [J].
BOWEN, WD ;
GENTLEMAN, S ;
HERKENHAM, M ;
PERT, CB .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (08) :4818-4822
[3]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[4]  
CHANG KJ, 1979, MOL PHARMACOL, V16, P91
[5]   REGIONAL DIFFERENCES IN MU-1-BINDING OF [3H][D-ALA2,D-LEU5]-ENKEPHALIN - COMPARISONS OF THALAMUS AND CORTEX IN THE RAT [J].
GOODMAN, RR ;
ADLER, BA ;
PASTERNAK, GW .
NEUROSCIENCE LETTERS, 1985, 59 (02) :155-158
[6]  
HAHN EF, 1982, J NEUROSCI, V2, P572
[7]   NALOXAZONE IRREVERSIBLY INHIBITS THE HIGH-AFFINITY BINDING OF [I-125]D-ALA2-D-LEU5-ENKEPHALIN [J].
HAZUM, E ;
CHANG, KJ ;
CUATRECASAS, P ;
PASTERNAK, GW .
LIFE SCIENCES, 1981, 28 (26) :2973-2979
[8]  
KENNER A, 1986, THESIS TEL AVIV U
[9]  
LING GSF, 1985, J PHARMACOL EXP THER, V232, P149
[10]   SEPARATION OF MORPHINE ANALGESIA FROM PHYSICAL-DEPENDENCE [J].
LING, GSF ;
MACLEOD, JM ;
LEE, S ;
LOCKHART, SH ;
PASTERNAK, GW .
SCIENCE, 1984, 226 (4673) :462-464