SYNTHESIS OF A GUANIDINO-SUGAR AS A GLYCOSYL CATION MIMIC

被引：26

作者：

FOTSCH, CH ^{[1
]}

WONG, CH ^{[1
]}

机构：

[1] Scripps Res Inst, DEPT CHEM, LA JOLLA, CA 92037 USA

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 21期

关键词：

D O I：

10.1016/S0040-4039(00)73215-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

?he synthesis of a guanidine threose (1a) is described. Under basic conditions, compound 1a equilibrates to tetrahydropyrimidine form 1b which acts as a transition-state inhibitor for green coffee bean galactosidase.

引用

页码：3481 / 3484

页数：4

共 23 条

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