SYNTHESIS AND STUDY OF A NON-MACROCYCLIC FK506 DERIVATIVE

被引：9

作者：

TEAGUE, SJ

COOPER, ME

DONALD, DK

FURBER, M

机构：

[1] Fisons plc, Pharmaceuticals Division, Loughborough, LE11 0RH, Bakewell Road

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1994年 / 4卷 / 13期

关键词：

D O I：

10.1016/S0960-894X(01)80570-9

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The affinity of a non macrocyclic analogue of FK506 for the immunophilin FKBP12 was The affinity of this analogue/FKBP12 complex for calcineurin was studied.

引用

页码：1581 / 1584

页数：4

共 27 条

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