POST-MODIFICATION OF PEPTOID SIDE-CHAINS - [3+2] CYCLOADDITION OF NITRILE OXIDES WITH ALKENES AND ALKYNES ON THE SOLID-PHASE

被引：54

作者：

PEI, YH ^{[1
]}

MOOS, WH ^{[1
]}

机构：

[1] CHIRON CORP,EMERYVILLE,CA 94608

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 32期

关键词：

CHEMICAL DIVERSITY; SOLID-PHASE SYNTHESIS; 3+2] CYCLOADDITION; NITRILE OXIDES; ISOXAZOLE; ISOXAZOLINE;

D O I：

10.1016/S0040-4039(00)78194-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of isoxazoles and isoxazolines were synthesized on solid-phase through [3+2] cycloaddition reactions of alkynes and alkenes with highly reactive nitrile oxides.

引用

页码：5825 / 5828

页数：4

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