AN EFFICIENT PARTIAL SYNTHESIS OF (+)-ARTEMISININ AND (+)-DEOXOARTEMISININ

被引：33

作者：

LANSBURY, PT

NOWAK, DM

机构：

[1] Department of Chemistry State University of New York at Buffalo, Buffalo

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 08期

关键词：

ARTEMISININ; DEOXOARTEMISININ; ARTEANNUIN B; ARTEANNUIC ACID; SINGLET OXYGEN; REDUCTIVE ELIMINATION; KETALIZATION; ALLYLIC OXIDATION;

D O I：

10.1016/S0040-4039(00)91851-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Arteannuic acid and arteannuin B are separately convertible into intermediate 8, which is transformed by four or five high-yielding steps into the title anti-malarial sesquiterpene peroxides.

引用

页码：1029 / 1032

页数：4

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