A GENERAL METHOD FOR COPPER-CATALYZED ARYLATION OF ACIDIC ARENE C-H BONDS. PREPARATION OF 2-CHLORO-5-(3-METHYLPHENYL)-THIOPHENE

被引：1

作者：

Alvarado, Joseph ^{[3
]}

Do, Hien-Quang ^{[3
,4
]}

Daugulis, Olafs ^{[1
,2
]}

Marsden, Peter C. ^{[5
]}

Ellman, Jonathan A.

机构：

[1] Univ Houston, Dept Chem, Houston, TX 77204 USA

[2] Univ Houston, Chem, Houston, TX 77204 USA

[3] Univ Houston, Houston, TX 77204 USA

[4] Univ Nat Sci, Ho Chi Minh City, Vietnam

[5] Pomona Coll, Claremont, CA 91711 USA

来源：

ORGANIC SYNTHESES | 2010年 / 87卷

关键词：

D O I：

10.15227/orgsyn.087.0184

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：184 / +

页数：10

共 10 条

[1] Direct palladium-catalyzed C-3 arylation of free (NH)-indoles with aryl bromides under ligandless conditions [J].

Bellina, Fabio ;

Benelli, Francesca ;

Rossi, Renzo .

JOURNAL OF ORGANIC CHEMISTRY, 2008, 73 (14) :5529-5535

[2] EQUILIBRIUM ACIDITIES IN DIMETHYL-SULFOXIDE SOLUTION [J].

BORDWELL, FG .

ACCOUNTS OF CHEMICAL RESEARCH, 1988, 21 (12) :456-463

[3] Palladium-Catalyzed Direct Arylation of Nitro-Substituted Aromatics with Aryl Halides [J].

Caron, Laurence ;

Campeau, Louis-Charles ;

Fagnou, Keith .

ORGANIC LETTERS, 2008, 10 (20) :4533-4536

[4] Palladium-catalyzed arylation of electron-rich heterocycles with aryl chlorides [J].

Chiong, Hendrich A. ;

Daugulis, Olafs .

ORGANIC LETTERS, 2007, 9 (08) :1449-1451

[5] A General Method for Copper-Catalyzed Arylation of Arene C-H Bonds [J].

Do, Hien-Ouang ;

Khan, Rana M. Kashif ;

Daugulis, Olafs .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2008, 130 (45) :15185-15192

[6] Copper-catalyzed arylation and alkenylation of polyfluoroarene C-H bonds [J].

Do, Hien-Quang ;

Daugulis, Olafs .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2008, 130 (04) :1128-+

[7] Formation of aryl-nitrogen, aryl-oxygen, and aryl-carbon bonds using well-defined copper(I)-based catalysts [J].

Gujadhur, RK ;

Bates, CG ;

Venkataraman, D .

ORGANIC LETTERS, 2001, 3 (26) :4315-4317

[8] An efficient copper-catalyzed coupling of aryl halides with imidazoles [J].

Kiyomori, A ;

Marcoux, JF ;

Buchwald, SL .

TETRAHEDRON LETTERS, 1999, 40 (14) :2657-2660

[9] Cu(II)-Catalyzed direct and site-selective arylation of indoles under mild conditions [J].

Phipps, Robert J. ;

Grimster, Neil P. ;

Gaunt, Matthew J. .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2008, 130 (26) :8172-+

[10] What are the pKa values of C-H bonds in aromatic heterocyclic compounds in DMSO? [J].

Shen, Kuang ;

Fu, Yao ;

Li, Jia-Ning ;

Liu, Lei ;

Guo, Qing-Xiang .

TETRAHEDRON, 2007, 63 (07) :1568-1576

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