SEQUENTIAL AND CASCADE [2+2]-CYCLOADDITION-PALLADIUM CATALYZED CYCLIZATION - BICYCLIC BETA-LACTAMS

被引：49

作者：

BURWOOD, M

DAVIES, B

DIAZ, I

GRIGG, R

MOLINA, P

SRIDHARAN, V

HUGHES, M

机构：

[1] UNIV LEEDS,SCH CHEM,LEEDS LS2 9JT,W YORKSHIRE,ENGLAND

[2] SMITHKLINE BEECHAM PHARMACEUT,HARLOW CM19 5AW,ESSEX,ENGLAND

[3] UNIV MURCIA,DEPT ORGAN CHEM,E-30071 MURCIA,SPAIN

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 49期

关键词：

D O I：

10.1016/0040-4039(95)01910-A

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Sequential and cascade ketene-imine [2+2]-cycloaddition-palladium catalysed cyclisation reactions occur in good yield. Racemic and homochiral examples incorporating a range of aromatic and heteroaromatic rings are reported.

引用

页码：9053 / 9056

页数：4

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