SYNTHESIS OF 13-EPI-TAXOL VIA A TRANSANNULAR DELIVERY OF A BOROHYDRIDE REAGENT

被引：21

作者：

HOEMANN, MZ ^{[1
]}

VANDERVELDE, D ^{[1
]}

GEORG, GI ^{[1
]}

JAYASINGHE, LR ^{[1
]}

机构：

[1] OREAD LABS,LAWRENCE,KS 66047

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1995年 / 60卷 / 09期

关键词：

D O I：

10.1021/jo00114a052

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：2918 / 2921

页数：4

共 48 条

[1] THE EFFECT OF THE AROMATIC RINGS OF TAXOL ON BIOLOGICAL-ACTIVITY AND SOLUTION CONFORMATION - SYNTHESIS AND EVALUATION OF SATURATED TAXOL AND TAXOTERE ANALOGS [J].

BOGE, TC ;

HIMES, RH ;

VANDERVELDE, DG ;

GEORG, GI .

JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (20) :3337-3343

[2] UNEXPECTEDLY FACILE HYDROLYSIS OF THE 2-BENZOATE GROUP OF TAXOL AND SYNTHESES OF ANALOGS WITH INCREASED ACTIVITIES [J].

CHAUDHARY, AG ;

GHARPURE, MM ;

RIMOLDI, JM ;

CHORDIA, MD ;

GUNATILAKA, AAL ;

KINGSTON, DGI ;

GROVER, S ;

LIN, CM ;

HAMEL, E .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1994, 116 (09) :4097-4098

[3] ON THE REACTION OF TAXOL WITH DAST [J].

CHEN, SH ;

HUANG, S ;

FARINA, V .

TETRAHEDRON LETTERS, 1994, 35 (01) :41-44

[4] FIRST SYNTHESES OF NOVEL PACLITAXEL(TAXOL) ANALOGS MODIFIED AT THE C4-POSITION [J].

CHEN, SH ;

KADOW, JF ;

FARINA, V ;

FAIRCHILD, CR ;

JOHNSTON, KA .

JOURNAL OF ORGANIC CHEMISTRY, 1994, 59 (21) :6156-6158

[5] STRUCTURE-ACTIVITY-RELATIONSHIPS OF TAXOL(R) - SYNTHESIS AND BIOLOGICAL EVALUATION OF C2 TAXOL ANALOGS [J].

CHEN, SH ;

FARINA, V ;

WEI, JM ;

LONG, B ;

FAIRCHILD, C ;

MAMBER, SW ;

KADOW, JF ;

VYAS, D ;

DOYLE, TW .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1994, 4 (03) :479-482

[6] SERENDIPITOUS SYNTHESIS OF A CYCLOPROPANE-CONTAINING TAXOL ANALOG VIA ANCHIMERIC PARTICIPATION OF AN UNACTIVATED ANGULAR METHYL-GROUP [J].

CHEN, SH ;

HUANG, S ;

WEI, JM ;

FARINA, V .

JOURNAL OF ORGANIC CHEMISTRY, 1993, 58 (17) :4520-4521

[7] SYNTHESIS OF 7-DEOXYTAXOL AND 7,10-DIDEOXYTAXOL VIA RADICAL INTERMEDIATES [J].

CHEN, SH ;

HUANG, S ;

KANT, J ;

FAIRCHILD, C ;

WEI, JM ;

FARINA, V .

JOURNAL OF ORGANIC CHEMISTRY, 1993, 58 (19) :5028-5029

[8] TAXOL STRUCTURE-ACTIVITY-RELATIONSHIPS - SYNTHESIS AND BIOLOGICAL EVALUATION OF 10-DEOXYTAXOL [J].

CHEN, SH ;

FAIRCHILD, C ;

MAMBER, SW ;

FARINA, V .

JOURNAL OF ORGANIC CHEMISTRY, 1993, 58 (11) :2927-2928

[9] SYNTHESIS AND BIOLOGICAL EVALUATION OF 4-DEACETOXYPACLITAXEL [J].

CHORDIA, MD ;

CHAUDHARY, AG ;

KINGSTON, DGI ;

JIANG, YQ ;

HAMEL, E .

TETRAHEDRON LETTERS, 1994, 35 (37) :6843-6846

[10] IMPROVED PROTECTION AND ESTERIFICATION OF A PRECURSOR OF THE TAXOTERE(R) AND TAXOL SIDE-CHAINS [J].

COMMERCON, A ;

BEZARD, D ;

BERNARD, F ;

BOURZAT, JD .

TETRAHEDRON LETTERS, 1992, 33 (36) :5185-5188

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