TAXOTERE(R) BY ESTERIFICATION WITH STEREOCHEMICALLY WRONG (2S,3S)-PHENYLISOSERINE DERIVATIVES

被引：37

作者：

DENIS, JN ^{[1
]}

KANAZAWA, AM ^{[1
]}

GREENE, AE ^{[1
]}

机构：

[1] UNIV JOSEPH FOURIER,LEDSS,F-38041 GRENOBLE,FRANCE

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 01期

关键词：

TAXOTERE(R); TAXOL; PHENYLISOSERINE; BACCATIN III;

D O I：

10.1016/0040-4039(94)88174-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Cyclically protected anti (2S, 3S) phenylisoserines on esterification with baccatin III derivatives afford Taxotere(R) and taxol precursors with the syn (2'R, 3'S) side chain.

引用

页码：105 / 108

页数：4

共 31 条

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[6] ASYMMETRIC-SYNTHESIS OF HOMOCHIRAL SYN-3-PHENYLISOSERINE AND ANTI-3-PHENYLISOSERINE DERIVATIVES - A PRACTICAL STRATEGY FOR THE SYNTHESIS OF THE TAXOL C-13 SIDE-CHAIN
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[8] CORRECTION
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[9] AN EFFICIENT, ENANTIOSELECTIVE SYNTHESIS OF THE TAXOL SIDE-CHAIN
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[10] AN IMPROVED SYNTHESIS OF THE TAXOL SIDE-CHAIN AND OF RP-56976
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[J]. JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (06) : 1957 - 1959

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