Heck reaction on solid support: Synthesis of indole analogs

被引：80

作者：

Yun, WY ^{[1
]}

Mohan, R ^{[1
]}

机构：

[1] BERLEX BIOSCI,RICHMOND,CA 94804

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 40期

关键词：

D O I：

10.1016/0040-4039(96)01635-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The intramolecular Heck reaction of polymer bound arylhalides such as 1 affords indole analogs 11 in high yield. The precursor is readily assembled from acid chlorides and allylic bromides and offers an approach to diverse libraries of indole analogs. Copyright (C) 1996 Elsevier Science Ltd

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页码：7189 / 7192

页数：4

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