Design and synthesis of conformationally constrained amino acids as versatile scaffolds and peptide mimetics

被引：783

作者：

Hanessian, S

McNaughtonSmith, G

Lombart, HG

Lubell, WD

机构：

[1] Département de Chimie, Université de Montréal, Montreal, Que. H3C 3J7, C.P. 6128, Succ. Centre-ville

[2] Parke-Davis Research Laboratories, Ann Arbor, MI

[3] ICAgen, Raleigh, NC

来源：

TETRAHEDRON | 1997年 / 53卷 / 38期

关键词：

D O I：

10.1016/S0040-4020(97)00476-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：12789 / 12854

页数：66

共 151 条

[1]

ADANG AEP, 1994, RECL TRAV CHIM PAY B, V113, P63

[2] ANTIBACTERIAL PROPERTIES OF THE BICYCLIC PYRAZOLIDINONES [J].

ALLEN, NE ;

HOBBS, JN ;

PRESTON, DA ;

TURNER, JR ;

WU, CYE .

JOURNAL OF ANTIBIOTICS, 1990, 43 (01) :92-99

[3] MOLECULAR MODELING OF GAMMA-LACTAM ANALOGS OF BETA-LACTAM ANTIBACTERIAL AGENTS - SYNTHESIS AND BIOLOGICAL EVALUATION OF SELECTED PENEM AND CARBAPENEM ANALOGS [J].

ALLEN, NE ;

BOYD, DB ;

CAMPBELL, JB ;

DEETER, JB ;

ELZEY, TK ;

FOSTER, BJ ;

HATFIELD, LD ;

HOBBS, JN ;

HORNBACK, WJ ;

HUNDEN, DC ;

JONES, ND ;

KINNICK, MD ;

MORIN, JM ;

MUNROE, JE ;

SWARTZENDRUBER, JK ;

VOGT, DG .

TETRAHEDRON, 1989, 45 (07) :1905-1928

[4] DESIGN OF ENZYME-INHIBITORS USING ITERATIVE PROTEIN CRYSTALLOGRAPHIC ANALYSIS [J].

APPELT, K ;

BACQUET, RJ ;

BARTLETT, CA ;

BOOTH, CLJ ;

FREER, ST ;

FUHRY, MAM ;

GEHRING, MR ;

HERRMANN, SM ;

HOWLAND, EF ;

JANSON, CA ;

JONES, TR ;

KAN, CC ;

KATHARDEKAR, V ;

LEWIS, KK ;

MARZONI, GP ;

MATTHEWS, DA ;

MOHR, C ;

MOOMAW, EW ;

MORSE, CA ;

OATLEY, SJ ;

OGDEN, RC ;

REDDY, MR ;

REICH, SH ;

SCHOETTLIN, WS ;

SMITH, WW ;

VARNEY, MD ;

VILLAFRANCA, JE ;

WARD, RW ;

WEBBER, S ;

WEBBER, SE ;

WELSH, KM ;

WHITE, J .

JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (07) :1925-1934

[5] THE DESIGN AND SYNTHESIS OF THE ANGIOTENSIN CONVERTING-ENZYME-INHIBITOR CILAZAPRIL AND RELATED BICYCLIC COMPOUNDS [J].

ATTWOOD, MR ;

HASSALL, CH ;

KROHN, A ;

LAWTON, G ;

REDSHAW, S .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1986, (06) :1011-1019

[6]

BACH AC, 1991, INT J PEPT PROT RES, V38, P314

[7] SYNTHESIS OF BICYCLIC GAMMA-LACTAMS VIA OXAZOLIDINONES [J].

BALDWIN, JE ;

LEE, E .

TETRAHEDRON, 1986, 42 (23) :6551-6554

[8]

BALDWIN JE, 1991, J ANTIBIOT, V44, P1

[9]

BALDWIN JE, 1992, HETEROCYCLES, V34, P903

[10] GAMMA-LACTAM FORMATION FROM TRIPEPTIDES WITH ISOPENICILLIN-N SYNTHASE [J].

BALDWIN, JE ;

NORRIS, WJ ;

FREEMAN, RT ;

BRADLEY, M ;

ADLINGTON, RM ;

LONGFOX, S ;

SCHOFIELD, CJ .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1988, (16) :1128-1130

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