Solid phase synthesis of urea libraries using a diversifiable thiophenoxy carbonyl linker

被引：40

作者：

Dressman, BA ^{[1
]}

Singh, U ^{[1
]}

Kaldor, SW ^{[1
]}

机构：

[1] Eli Lilly & Co, Lilly Res Lab, Lilly Corp Ctr, Indianapolis, IN 46285 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 22期

关键词：

D O I：

10.1016/S0040-4039(98)00652-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A method for the solid phase synthesis of urea libraries from primary and secondary amines is described which utilizes a thiophenoxy carbonyl linker. Sequential release of different urea products from a common batch of resin using a "milking" procedure has also been accomplished. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：3631 / 3634

页数：4

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