Highly efficient synthesis of pyrimidines under microwave-assisted conditions

被引：72

作者：

Bagley, MC ^{[1
]}

Hughes, DD ^{[1
]}

Taylor, PH ^{[1
]}

机构：

[1] Cardiff Univ, Dept Chem, Cardiff CF10 3TB, S Glam, Wales

来源：

SYNLETT | 2003年 / 02期

关键词：

pyrimidines; microwave synthesis; heterocycles;

D O I：

10.1055/s-2003-36781

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Microwave irradiation of an amidine and alkynone in acetonitrile at 120 degreesC dives 2,4-disubstituted and 2,4,6-trisubstituted pyrimidines in very high yield.

引用

页码：259 / 261

页数：3

共 27 条

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