Solid phase synthesis of aspartyl peptide aldehydes

被引：9

作者：

Tong, XH ^{[1
]}

Hong, A ^{[1
]}

机构：

[1] AnaSpec Inc, San Jose, CA 95131 USA

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 46期

关键词：

D O I：

10.1016/S0040-4039(00)01615-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient method for the solid phase synthesis of aspartyl aldehyde peptides has been developed. It uses a low cost synthetic process for the preparation of Fmoc-protected Weinreb amide linker. This procedure covers several tetrapeptide aspartyl aldehydes as well as biotinylated tetrapeptide aspartyl aldehydes. (C) 2000 Elsevier Science Ltd. All rights reserved.

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页码：8857 / 8860

页数：4

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