Solution-phase parallel synthesis of benzoxazines using a polymer-supported carbodiimide

被引：15

作者：

Buckman, BO ^{[1
]}

Morrissey, MM ^{[1
]}

Mohan, R ^{[1
]}

机构：

[1] Berlex Biosci, Pharmaceut Discovery, Richmond, CA 94804 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(98)00012-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A diverse library of 2-aminobenzoxazines 3 has been synthesized using a two step approach. Addition of anthranilic acids to isocyanates affords ureas 2 that can be cyclized by polymer-supported EDC to give 2-aminobenzoxazines 3. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：1487 / 1488

页数：2

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