Optimisation and synthesis of libraries derived from phenolic amino acid scaffolds

被引：11

作者：

Morley, AD ^{[1
]}

机构：

[1] Aventis Pharma Ltd, Dagenham RM10 7XS, Essex, England

来源：

TETRAHEDRON LETTERS | 2000年 / 41卷 / 38期

关键词：

solid-phase synthesis; Mitsunobu reactions; acylation; reductive amination;

D O I：

10.1016/S0040-4039(00)01264-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Functionalisation of a series of resin bound phenolic amino acids is described, employing Irori technology to produce multidimensional libraries. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

收藏

页码：7405 / 7408

页数：4

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